SCHEMBL17864639

SCHEMBL17864639

C/C(=N\O)c1cc2c(C)ccc(C)c2o1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
RARA P10276 14/20 0.36
RARB P10826 14/20 0.36
RARG P13631 14/20 0.36
GPR55 Q9Y2T6 2/20 0.33
HSD17B10 Q99714 1/20 0.33
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19599548 0.81 LMNA (0.37) RARARARBRARGGPR55CNR2
SCHEMBL17843543 0.81 LMNA (0.37) RARARARBRARGGPR55CNR2
SCHEMBL17864569 0.81 LMNA (0.37) RARARARBRARGGPR55CNR2
SCHEMBL17843583 0.74 RARA (0.50) KDM4ERARARARBRARG
SCHEMBL29396158 0.73 RARA (0.43) RARARARBRARG
SCHEMBL21562101 0.73 RARA (0.43) RARARARBRARG
SCHEMBL17988331 0.71 NPC1 (0.40) KDM4EHSD17B10
SCHEMBL23691679 0.70 MAPT (0.49) KDM4ERARARARBRARGGPR55
SCHEMBL19583279 0.70 RARA (0.36) RARARARBRARGGPR55CNR2
SCHEMBL17864618 0.69 RARA (0.37) KDM4ERARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016097004-A1 BICYCLOHETEROARYL-HETEROARYL-BENZOIC ACID COMPOUNDS AS RETINOIC ACID RECEPTOR BETA (RARβ) AGONISTS KING'S COLLEGE LONDON (GB) 2016-06-23 WO disclosed