SCHEMBL17865741

SCHEMBL17865741

C[C@@H](C(=O)N1CCN(C(=O)OC(C)(C)C)CC1)[C@H]1NC(=O)[C@H]1CCO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 2/20 0.42
CRBN Q96SW2 2/20 0.42
ADAM17 P78536 2/20 0.41
MMP3 P08254 1/20 0.41
HTT P42858 2/20 0.41
ATM Q13315 1/20 0.41
MAPT P10636 2/20 0.38
MAPK1 P28482 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 2/20 0.37
THRB P10828 1/20 0.37
TPSAB1 Q15661 3/20 0.37
TPSD1 Q9BZJ3 3/20 0.37
TPSG1 Q9NRR2 3/20 0.37
DTYMK P23919 1/20 0.36
MMP13 P45452 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17865749 1.00 DDB1 (0.42) DDB1CRBNADAM17MMP3HTT
SCHEMBL19521198 0.82 HTT (0.35) ADAM17MMP3HTTNPC1ALDH1A1
SCHEMBL19521178 0.81 ALDH1A1 (0.44) MAPTNPC1ALDH1A1RAB9AKDM4E
SCHEMBL17865738 0.80 HTT (0.43) DDB1CRBNADAM17MMP3HTT
SCHEMBL20153494 0.80 HTT (0.43) DDB1CRBNADAM17MMP3HTT
SCHEMBL17865748 0.80 HTT (0.43) DDB1CRBNADAM17MMP3HTT
SCHEMBL17865739 0.80 HTT (0.43) DDB1CRBNADAM17MMP3HTT
SCHEMBL19521241 0.74 HRH4 (0.30)
SCHEMBL19521177 0.73 ADAMTS5 (0.48) ADAMTS5
SCHEMBL20168992 0.72 MMP2 (0.32) ADAM17ADAMTS5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3036219-A2 NOVEL BETA LACTAMS AS MODULATORS OF GLUTAMATE UPTAKE AND METHODS FOR USE THEREOF Temple University Of The Commonwealth System Of Higher Education (US) 2016-06-29 EP claimed