SCHEMBL17896604

SCHEMBL17896604

Cc1ccncc1-c1nc2cc(F)cc(F)c2n1C

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 11/20 0.53
CYP11B2 P19099 4/20 0.48
CYP11B1 P15538 3/20 0.48
PDE2A O00408 6/20 0.44
CYP17A1 P05093 2/20 0.42
CYP1A2 P05177 1/20 0.40
TDO2 P48775 1/20 0.39
PTGS2 P35354 1/20 0.38
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460559 0.81 CYP11B2 (0.46) PDE10ACYP11B2CYP11B1PDE2A
SCHEMBL17883780 0.81 CYP11B2 (0.68) CYP11B2CYP11B1CYP17A1CYP1A2
SCHEMBL463351 0.80 CYP11B2 (0.67) PDE10ACYP11B2CYP11B1PDE2ACYP17A1
SCHEMBL17896700 0.78 CYP11B2 (0.62) CYP11B2CYP11B1
SCHEMBL17896602 0.78 CYP11B2 (0.67) PDE10ACYP11B2CYP11B1PDE2APOLB
SCHEMBL432104 0.77 PDE10A (0.65) PDE10ACYP11B2CYP11B1PDE2ATDO2
SCHEMBL17896600 0.73 CYP11B2 (0.45) CYP11B2CYP11B1CYP1A2
SCHEMBL17896702 0.72 CYP11B2 (0.41) PDE10ACYP11B2CYP11B1PDE2ATDO2
SCHEMBL17896699 0.70 PTGS2 (0.39) CYP11B2CYP11B1PTGS2
SCHEMBL461417 0.69 PDE10A (0.46) PDE10ACYP11B2CYP11B1PDE2ACYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed