SCHEMBL10175342

SCHEMBL10175342

Cn1c(-c2cncc(Br)c2)nc2cc(C#N)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.46
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP11B1 P15538 6/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
PTGER4 P35408 1/20 0.37
ATM Q13315 1/20 0.37
PTGS2 P35354 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896613 0.90 CYP11B2 (0.46) CYP11B2CYP11B1
SCHEMBL10175348 0.87 CYP11B2 (0.48) CYP11B2ALDH1A1CYP11B1KDM4EGLA
SCHEMBL17896641 0.85 CYP11B2 (0.47) CYP11B2ALDH1A1CYP11B1KDM4EGLA
SCHEMBL17896642 0.83 ALOX5AP (0.46) CYP11B2CYP11B1PTGER4PTGS2CA12
SCHEMBL17883795 0.82 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL10175125 0.82 CYP11B2 (0.70) CYP11B2CYP11B1
SCHEMBL10175439 0.81 CYP11B2 (0.46) CYP11B2CYP11B1ATM
SCHEMBL4243953 0.81 CYP11B2 (0.69) CYP11B2CYP11B1ATMPTGS2
SCHEMBL10175456 0.80 MEN1 (0.57) CYP11B2ALDH1A1NPC1TP53MAPT
SCHEMBL13749911 0.79 ATM (0.52) CYP11B2ALDH1A1NPC1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed