SCHEMBL17896641

SCHEMBL17896641

Cn1c(-c2cncc(F)c2)nc2cc(C#N)ccc21

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 13/20 0.47
CYP11B1 P15538 11/20 0.47
CYP19A1 P11511 1/20 0.43
ADRA2B P18089 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
TLR7 Q9NYK1 1/20 0.39
PTGER4 P35408 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896612 0.90 CYP11B2 (0.52) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL10175348 0.87 CYP11B2 (0.48) CYP11B2CYP11B1KDM4EALDH1A1GLA
SCHEMBL10175342 0.85 CYP11B2 (0.46) CYP11B2CYP11B1KDM4EALDH1A1GLA
SCHEMBL17883795 0.84 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL17896718 0.84 CYP11B2 (0.56) CYP11B2CYP11B1CYP19A1ADRA2BATM
SCHEMBL17896642 0.83 ALOX5AP (0.46) CYP11B2CYP11B1PTGER4
SCHEMBL17896644 0.82 CYP11B2 (0.71) CYP11B2CYP11B1CYP19A1ADRA2B
SCHEMBL10175439 0.81 CYP11B2 (0.46) CYP11B2CYP11B1ATM
SCHEMBL4243953 0.81 CYP11B2 (0.69) CYP11B2CYP11B1CYP19A1ATM
SCHEMBL17896665 0.81 KDM4E (0.52) CYP11B2CYP11B1CYP19A1ADRA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed