SCHEMBL10175348

SCHEMBL10175348

Cc1cncc(-c2nc3cc(C#N)ccc3n2C)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 11/20 0.48
CYP11B1 P15538 8/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
ATM Q13315 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
PTGER4 P35408 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175107 0.90 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL10175342 0.87 CYP11B2 (0.46) CYP11B2CYP11B1KDM4EALDH1A1GLA
SCHEMBL17896641 0.87 CYP11B2 (0.47) CYP11B2CYP11B1KDM4EALDH1A1GLA
SCHEMBL17896642 0.85 ALOX5AP (0.46) CYP11B2CYP11B1CA12CA1CA2
SCHEMBL17883795 0.84 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL10175439 0.83 CYP11B2 (0.46) CYP11B2CYP11B1ATM
SCHEMBL4243953 0.83 CYP11B2 (0.69) CYP11B2CYP11B1ATM
SCHEMBL10175456 0.82 MEN1 (0.57) CYP11B2CYP11B1KDM4EALDH1A1GLA
SCHEMBL13749911 0.81 ATM (0.52) CYP11B2KDM4EALDH1A1GLAGAA
SCHEMBL10175442 0.81 BRD4 (0.46) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed