SCHEMBL17896743

SCHEMBL17896743

Cn1c(-c2cncc3ccccc23)nc2cc(F)c(Cl)cc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 17/20 0.60
CYP11B1 P15538 12/20 0.42
CYP17A1 P05093 2/20 0.39
CYP3A4 P08684 1/20 0.38
ERN1 O75460 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
RAB9A P51151 1/20 0.37
NFKB2 Q00653 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896648 0.84 CYP11B2 (0.59) CYP11B2CYP11B1CYP3A4ERN1KDM4E
SCHEMBL459587 0.81 CYP11B2 (0.63) CYP11B2CYP11B1CYP3A4
SCHEMBL17896741 0.81 CYP11B2 (0.47) CYP11B2CYP11B1CYP17A1KDM4EALDH1A1
SCHEMBL17896744 0.81 CYP11B2 (0.47) CYP11B2CYP11B1CYP17A1CYP3A4KDM4E
SCHEMBL432410 0.79 CYP11B2 (0.56) CYP11B2CYP11B1ALDH1A1SMN1; SMN2
SCHEMBL434081 0.78 CYP11B2 (0.53) CYP11B2CYP11B1CYP3A4KDM4EALDH1A1
SCHEMBL10175154 0.77 MEN1 (0.54) CYP11B2CYP11B1KDM4EALDH1A1LMNA
SCHEMBL17883780 0.77 CYP11B2 (0.68) CYP11B2CYP11B1CYP17A1CYP3A4ERN1
SCHEMBL460601 0.76 CYP11B2 (0.67) CYP11B2CYP11B1CYP3A4ERN1
SCHEMBL17896589 0.76 CYP11B2 (0.51) CYP11B2CYP11B1CYP3A4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed