SCHEMBL434081

SCHEMBL434081

Cn1c(-c2cncc3ccccc23)nc2cc(Br)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.53
RAB9A P51151 5/20 0.49
NPC1 O15118 4/20 0.49
MAPT P10636 3/20 0.49
TP53 P04637 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
ALDH1A1 P00352 3/20 0.49
TSHR P16473 2/20 0.49
ALOX15 P16050 1/20 0.49
MAPK1 P28482 1/20 0.49
ATM Q13315 1/20 0.41
CYP11B1 P15538 5/20 0.40
PTGER4 P35408 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CASP1 P29466 1/20 0.40
POLB P06746 1/20 0.39
KDM4E B2RXH2 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17896620 0.84 SMN1; SMN2 (0.46) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL17896761 0.82 CYP11B2 (0.56) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL22439775 0.82 ALDH1A1 (0.60) RAB9ANPC1MAPTTP53SMN1; SMN2
SCHEMBL10175444 0.81 CYP11B2 (0.50) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL17896648 0.81 CYP11B2 (0.59) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL17896763 0.80 CYP11B2 (0.48) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL17883791 0.79 CYP11B2 (0.47) CYP11B2CYP11B1
SCHEMBL17896743 0.78 CYP11B2 (0.60) CYP11B2RAB9ANPC1MAPTTP53
SCHEMBL17896738 0.77 BRD4 (0.54) CYP11B2
SCHEMBL30663907 0.76 RAB9A (0.53) RAB9ANPC1MAPTTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP disclosed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO disclosed