SCHEMBL460601

SCHEMBL460601

Cn1c(-c2cncc3ccccc23)nc2c(F)c(F)ccc21

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 15/20 0.67
CYP11B1 P15538 12/20 0.43
ERN1 O75460 1/20 0.40
PRKCZ Q05513 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
TLR7 Q9NYK1 1/20 0.36
PIK3CD O00329 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL460502 0.85 CYP11B2 (0.56) CYP11B2CYP11B1ERN1PRKCZ
SCHEMBL10175445 0.81 CYP11B2 (1.00) CYP11B2CYP11B1ERN1PRKCZCNR1
SCHEMBL461417 0.80 PDE10A (0.46) CYP11B2CYP11B1CYP1A2
SCHEMBL17896743 0.76 CYP11B2 (0.60) CYP11B2CYP11B1ERN1CYP3A4
SCHEMBL17896648 0.75 CYP11B2 (0.59) CYP11B2CYP11B1ERN1CYP1A2CYP3A4
SCHEMBL463000 0.73 CYP11B2 (0.41) CYP11B2CYP11B1TLR7
SCHEMBL434081 0.73 CYP11B2 (0.53) CYP11B2CYP11B1PRKCZCNR1CNR2
SCHEMBL17883780 0.72 CYP11B2 (0.68) CYP11B2CYP11B1ERN1PRKCZCNR1
SCHEMBL17896761 0.71 CYP11B2 (0.56) CYP11B2CYP11B1ERN1CYP1A2CYP3A4
SCHEMBL10175444 0.70 CYP11B2 (0.50) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP claimed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO claimed