SCHEMBL17897154

SCHEMBL17897154

c1ccc2c(c1)ncc1n[nH]nc12

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
KDM4E B2RXH2 1/20 0.45
GPR3 P46089 1/20 0.45
ADORA3 P0DMS8 1/20 0.40
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
TLR7 Q9NYK1 1/20 0.38
PDPK1 O15530 1/20 0.37
CA12 O43570 1/20 0.37
PARP1 P09874 1/20 0.37
ALOX15 P16050 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CA9 Q16790 1/20 0.37
TNKS2 Q9H2K2 1/20 0.37
ERN1 O75460 1/20 0.37
TOP2A P11388 1/20 0.37
TDO2 P48775 2/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3857012 0.71 TSHR (0.48) TSHRKEAP1NFE2L2SMN1; SMN2TDO2
SCHEMBL27727935 0.71 KDM4E (0.59) KDM4EGPR3ADORA3TLR7SMN1; SMN2
SCHEMBL17917460 0.71 LMNA (0.48) KDM4EGPR3ADORA3TLR7ERN1
Benzotriazole SCHEMBL29355833 0.69 TSHR (1.00) TSHRKDM4EGPR3KEAP1NFE2L2
Benzotriazole SCHEMBL171464 0.69
SCHEMBL1727666 0.69 KDM4E (0.52) KDM4EGPR3ADORA3TLR7PDPK1
SCHEMBL30951595 0.69 KDM4E (0.52) KDM4EGPR3ADORA3TLR7PDPK1
SCHEMBL2363194 0.68 KDM4E (0.50) TSHRKDM4EGPR3ADORA3TLR7
SCHEMBL253096 0.68 GPR3 (0.50) KDM4EGPR3PDPK1CA12PARP1
SCHEMBL30539895 0.68 GPR3 (0.50) KDM4EGPR3PDPK1CA12PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160197275-A1 EMITTER HAVING A CONDENSED RING SYSTEM MERCK PATENT GMBH (DE) 2016-07-07 US disclosed
US-20160197275-A1 EMITTER HAVING A CONDENSED RING SYSTEM MERCK PATENT GMBH (DE) 2016-07-07 US disclosed