SCHEMBL17898107

SCHEMBL17898107

NS(=O)(=O)OC[C@H]1C[C@@H](n2cnc3c(NCc4ccccc4)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 5/20 0.60
NAE1 Q13564 3/20 0.53
UBA3 Q8TBC4 3/20 0.53
DNPH1 O43598 1/20 0.52
CA2 P00918 1/20 0.52
TP53 P04637 1/20 0.51
SLC29A1 Q99808 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
NT5E P21589 1/20 0.49
P2RX3 P56373 1/20 0.49
P2RX2 Q9UBL9 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1795319 0.84 CA2 (0.55) NAE1UBA3CA2
SCHEMBL23080273 0.84 CA2 (0.55) NAE1UBA3CA2
SCHEMBL17875220 0.83 SLC29A1 (0.60) ADORA3NAE1UBA3DNPH1TP53
SCHEMBL10186161 0.83 SLC29A1 (0.60) ADORA3NAE1UBA3DNPH1TP53
SCHEMBL1796246 0.83 SLC29A1 (0.60) ADORA3NAE1UBA3DNPH1TP53
SCHEMBL12566881 0.83 CA2 (0.53) NAE1UBA3DNPH1CA2
SCHEMBL17889870 0.82 DNPH1 (0.75) ADORA3NAE1UBA3DNPH1TP53
SCHEMBL1796735 0.82 DNPH1 (0.75) ADORA3NAE1UBA3DNPH1TP53
SCHEMBL1795912 0.81 ADORA3 (0.63) ADORA3DNPH1TP53SLC29A1TDP1
SCHEMBL1949613 0.80 DNPH1 (0.65) ADORA3NAE1UBA3DNPH1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170073367-A9 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES MILLENIUM PHARMACEUTICALS, INC. 2017-03-16 US disclosed
US-20170073367-A9 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES MILLENIUM PHARMACEUTICALS, INC. 2017-03-16 US disclosed
US-20160194348-A1 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES MILLENNIUM PHARM INC (US) 2016-07-07 US disclosed
US-20160194348-A1 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES MILLENNIUM PHARM INC (US) 2016-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170073367-A9 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES TYMP, TYMS, PPA1 ADORA3 1669/4885NAE1 257/4885UBA3 235/4885
US-20160194348-A1 SUBSTITUTED PYRROLO[2,3-D]PYRIMIDINES TYMP, TYMS, PPA1 ADORA3 1669/4885NAE1 257/4885UBA3 235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.