SCHEMBL179049

SCHEMBL179049

Cc1ccc(S(=O)(=O)OCC(F)COS(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGER Q15109 1/20 0.44
VDR P11473 1/20 0.44
GAA P10253 2/20 0.43
STAT3 P40763 1/20 0.42
ALDH1A1 P00352 4/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA1 P00915 3/20 0.41
CA9 Q16790 3/20 0.41
CA12 O43570 2/20 0.41
CA2 P00918 2/20 0.41
CA3 P07451 1/20 0.41
CA6 P23280 1/20 0.41
CA5A P35218 1/20 0.41
CA7 P43166 1/20 0.41
CA5B Q9Y2D0 1/20 0.41
DHODH Q02127 1/20 0.40
TLR9 Q9NR96 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10339892 0.93 ALDH1A1 (0.41) AGERVDRGAASTAT3ALDH1A1
SCHEMBL116604 0.91 AGER (0.41) AGERVDRGAASTAT3ALDH1A1
SCHEMBL25345480 0.91 AGER (0.41) AGERVDRGAASTAT3ALDH1A1
SCHEMBL30802773 0.91 AGER (0.41) AGERVDRGAASTAT3ALDH1A1
SCHEMBL116676 0.91 AGER (0.41) AGERVDRGAASTAT3ALDH1A1
SCHEMBL17396769 0.90 CA12 (0.40) AGERVDRGAASTAT3ALDH1A1
SCHEMBL28655071 0.90 DHODH (0.42) AGERVDRGAASTAT3ALDH1A1
SCHEMBL17396847 0.90 CA12 (0.40) AGERVDRGAASTAT3ALDH1A1
SCHEMBL336511 0.89 AGER (0.44) AGERVDRGAASTAT3ALDH1A1
SCHEMBL17427977 0.89 CA12 (0.45) AGERVDRGAASTAT3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12358929-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2025-07-15 US disclosed
US-20240294546-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2024-09-05 US disclosed
EP-3558318-B1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2023-12-20 EP disclosed
US-11807650-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2023-11-07 US disclosed
US-11807650-B2 NMDA receptor modulators and uses thereof NOVARTIS AG (CH) 2023-11-07 US disclosed
US-11679095-B2 Macrophages/microglia in neuro-inflammation associated with neurodegenerative diseases THE GENERAL HOSPITAL CORPORATION (US) 2023-06-20 US disclosed
US-20220153755-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2022-05-19 US disclosed
US-11274107-B2 NMDA receptor modulators and uses thereof CADENT THERAPEUTICS, INC. (US) 2022-03-15 US disclosed
US-10738063-B2 6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-carboxamide compounds PFIZER INC. (US) 2020-08-11 US disclosed
US-20200087323-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF NOVARTIS AG (CH) 2020-03-19 US disclosed
US-20160263257-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT THE GENERAL HOSPITAL CORPORATION 2016-09-15 US disclosed
EP-2944637-A1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM Corporation (JP) 2015-11-18 EP disclosed
EP-2944637-A1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF FUJIFILM Corporation (JP) 2015-11-18 EP disclosed
WO-2014109414-A1 NITROGEN-CONTAINING HETEROCYLIC COMPOUND OR SALT THEREOF 富士フイルム株式会社 (JP) 2014-07-17 WO disclosed
US-20140140927-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT THE GENERAL HOSPITAL CORPORATION (US) 2014-05-22 US disclosed
US-20120058049-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT THE GENERAL HOSPITAL CORPORATION 2012-03-08 US disclosed
WO-2010088455-A2 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT THE GENERAL HOSPITAL CORPORATION (US) 2010-08-05 WO disclosed
US-20090227616-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION, A CORPORATION 2009-09-10 US disclosed
EP-1948185-A2 INHIBITORS OF AKT ACTIVITY SmithKline Beecham Corporation (US) 2008-07-30 EP disclosed
WO-2007058852-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2007-05-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090227616-A1 INHIBITORS OF AKT ACTIVITY PI4KB, PIK3CA, AKT2 AGER 4297/4885VDR 4415/4885GAA 2624/4885
US-11807650-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-11274107-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-10738063-B2 6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-2-carboxamide compounds PDE4B, PDE5A, PDE3B AGER 3434/4885VDR 3589/4885GAA 1441/4885
US-20240294546-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-11679095-B2 Macrophages/microglia in neuro-inflammation associated with neurodegenerative diseases CD68, PRNP, HTT AGER 1155/4885VDR 4264/4885GAA 613/4885
US-12358929-B2 NMDA receptor modulators and uses thereof GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-20140140927-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT PSEN1, PSEN2, CROCC AGER 359/4885VDR 1549/4885GAA 1525/4885
US-20160263257-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT PSEN1, CROCC, PSEN2 AGER 337/4885VDR 1711/4885GAA 1408/4885
US-20200087323-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-20220153755-A1 NMDA RECEPTOR MODULATORS AND USES THEREOF GRIN1, GRIN2A, GRIN2C AGER 684/4885VDR 289/4885GAA 3389/4885
US-20120058049-A1 CROMOLYN DERIVATIVES AND RELATED METHODS OF IMAGING AND TREATMENT CLN6, CA6, GALNT6 AGER 747/4885VDR 2128/4885GAA 2158/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.