SCHEMBL17907952

SCHEMBL17907952

COc1ccc2c(c1)cc1n2CC(N(C)Cc2ccccc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
KMT2A Q03164 1/20 0.39
GRIN2B Q13224 1/20 0.39
HTR6 P50406 2/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.38
CLK1 P49759 1/20 0.38
DYRK1A Q13627 1/20 0.38
GRIK1 P39086 1/20 0.37
GRIK2 Q13002 1/20 0.37
HTR1A P08908 1/20 0.36
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907919 0.88 PTGDR2 (0.41) GRIN2BPTGDR2
SCHEMBL17907987 0.86 GRIN2B (0.41) KMT2AGRIN2BMAPTPTGDR2
SCHEMBL17907982 0.85 GRIN2B (0.44) HTR2AHTR2CGRIN2BPTGDR2SLC6A4
SCHEMBL17908006 0.85 NOS3 (0.41) HTR2AHTR2CKMT2AGRIN2BKDM4E
SCHEMBL17907957 0.85 CYP2D6 (0.42) KMT2AGRIN2BPTGDR2
SCHEMBL17907929 0.78 CYP2D6 (0.42) KMT2AGRIN2BPTGDR2
SCHEMBL17907974 0.78 NOS3 (0.41) HTR2AHTR2CGRIN2BPTGDR2SLC6A4
SCHEMBL17908001 0.77 MAOA (0.47) ALDH1A1HTR2AHTR2CMAOAMAOB
SCHEMBL17907936 0.77 GRIN2B (0.39) GRIN2BHTR6PTGDR2
SCHEMBL17907970 0.73 PTGDR2 (0.49) ALDH1A1KMT2AHTR6POLBPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed