SCHEMBL17907957

SCHEMBL17907957

CN(Cc1ccccc1)C1CCc2cc3cc(F)ccc3n2C1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
CHRM1 P11229 1/20 0.42
HRH1 P35367 1/20 0.42
GRIN2B Q13224 1/20 0.40
PTGDR2 Q9Y5Y4 9/20 0.38
KMT2A Q03164 1/20 0.36
CCR3 P51677 1/20 0.36
TBXA2R P21731 1/20 0.36
PTGDR Q13258 1/20 0.36
NAAA Q02083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907929 0.91 CYP2D6 (0.42) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17907987 0.88 GRIN2B (0.41) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17907982 0.87 GRIN2B (0.44) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17908006 0.87 NOS3 (0.41) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17907952 0.85 ALDH1A1 (0.41) GRIN2BPTGDR2KMT2A
SCHEMBL17907919 0.83 PTGDR2 (0.41) GRIN2BPTGDR2
SCHEMBL17907936 0.81 GRIN2B (0.39) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17907974 0.80 NOS3 (0.41) CYP2D6CHRM1HRH1GRIN2BPTGDR2
SCHEMBL17907975 0.75 CCR3 (0.50) GRIN2BCCR3
SCHEMBL17907943 0.71 PTGDR2 (0.59) PTGDR2TBXA2RPTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed