SCHEMBL17907987

SCHEMBL17907987

Cc1ccc2c(c1)cc1n2CC(N(C)Cc2ccccc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.41
OPRM1 P35372 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
NAAA Q02083 2/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TSHR P16473 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
AGTR2 P50052 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP2D6 P10635 1/20 0.35
CHRM1 P11229 1/20 0.35
HRH1 P35367 1/20 0.35
SLC18A3 Q16572 1/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
MEN1 O00255 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907982 0.88 GRIN2B (0.44) GRIN2BOPRM1SIGMAR1NAAAJAK2
SCHEMBL17908006 0.88 NOS3 (0.41) GRIN2BOPRM1SIGMAR1NAAAPTGDR2
SCHEMBL17907957 0.88 CYP2D6 (0.42) GRIN2BNAAAPTGDR2KMT2ACYP2D6
SCHEMBL17907952 0.86 ALDH1A1 (0.41) GRIN2BPTGDR2KMT2AMAPT
SCHEMBL17907919 0.82 PTGDR2 (0.41) GRIN2BJAK2JAK1PTGDR2
SCHEMBL17907974 0.81 NOS3 (0.41) GRIN2BNAAAPTGDR2CYP2D6CHRM1
SCHEMBL17907929 0.81 CYP2D6 (0.42) GRIN2BNAAAPTGDR2KMT2ACYP2D6
SCHEMBL17907936 0.79 GRIN2B (0.39) GRIN2BOPRM1SIGMAR1NAAAJAK2
SCHEMBL17907992 0.76 ACHE (0.48) GRIN2BKMT2AMEN1L3MBTL1
SCHEMBL17907921 0.70 PTGDR2 (0.46) PTGDR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed