SCHEMBL17907992

SCHEMBL17907992

Cc1ccc2c(c1)cc1n2CC(NCc2ccccc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 0.48
BACE1 P56817 7/20 0.48
BCHE P06276 6/20 0.48
RB1 P06400 4/20 0.47
GRIN2B Q13224 4/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
EBP Q15125 1/20 0.40
DHCR7 Q9UBM7 1/20 0.40
TACR1 P25103 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13279646 0.87 GRIN2B (0.49) ACHEBACE1BCHERB1GRIN2B
SCHEMBL17907975 0.86 CCR3 (0.50) ACHEBACE1BCHEGRIN2B
SCHEMBL17907942 0.86 BCHE (0.49) ACHEBACE1BCHEGRIN2BMEN1
SCHEMBL17908001 0.85 MAOA (0.47) ACHEBACE1BCHEGRIN2BMEN1
SCHEMBL17907961 0.81 BCHE (0.53) ACHEBACE1BCHEGRIN2B
SCHEMBL17907977 0.79 CCR3 (0.50) ACHEBACE1BCHEGRIN2B
SCHEMBL17907991 0.79 BCHE (0.49) ACHEBACE1BCHEGRIN2BMEN1
SCHEMBL17907999 0.76 BCHE (0.51) ACHEBACE1BCHEGRIN2B
SCHEMBL6337839 0.69 GRIN2B (0.71) ACHEBACE1RB1GRIN2B
SCHEMBL18828833 0.65 LTA4H (0.63) ACHEBACE1BCHERB1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed