SCHEMBL17907975

SCHEMBL17907975

Fc1ccc2c(c1)cc1n2CC(NCc2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 1/20 0.50
BCHE P06276 9/20 0.48
ACHE P22303 9/20 0.48
BACE1 P56817 9/20 0.48
GRIN2B Q13224 4/20 0.44
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17907977 0.91 CCR3 (0.50) CCR3BCHEACHEBACE1GRIN2B
SCHEMBL13279646 0.87 GRIN2B (0.49) BCHEACHEBACE1GRIN2BDRD2
SCHEMBL17907942 0.86 BCHE (0.49) CCR3BCHEACHEBACE1GRIN2B
SCHEMBL17907992 0.86 ACHE (0.48) BCHEACHEBACE1GRIN2B
SCHEMBL17908001 0.83 MAOA (0.47) BCHEACHEBACE1GRIN2BDRD2
SCHEMBL17907961 0.83 BCHE (0.53) CCR3BCHEACHEBACE1GRIN2B
SCHEMBL17907991 0.79 BCHE (0.49) CCR3BCHEACHEBACE1GRIN2B
SCHEMBL17907999 0.79 BCHE (0.51) CCR3BCHEACHEBACE1GRIN2B
SCHEMBL17907957 0.75 CYP2D6 (0.42) CCR3GRIN2B
SCHEMBL12347570 0.69 TBXA2R (0.55) CCR3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2697223-B1 7-(HETEROARYL-AMINO)-6,7,8,9-TETRAHYDROPYRIDO[1,2-A]INDOL ACETIC ACID DERIVATIVES AND THEIR USE AS PROSTAGLANDIN D2 RECEPTOR MODULATORS ACTELION PHARMACEUTICALS LTD (CH) 2016-07-13 EP disclosed