SCHEMBL1795182

SCHEMBL1795182

Cc1cc(NC(=O)c2nc(C)cc(-c3ccc(F)c(Cl)c3)c2C)ccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.50
SORT1 Q99523 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
SMARCA2 P51531 1/20 0.44
SMARCA4 P51532 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KMO O15229 1/20 0.43
ATR Q13535 1/20 0.43
HDAC4 P56524 1/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
MAPK1 P28482 1/20 0.41
LMNA P02545 1/20 0.40
KDR P35968 1/20 0.40
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794085 0.84 GRM5 (0.54) GRM5SORT1SMARCA2SMARCA4MEN1
SCHEMBL1795467 0.82 SORT1 (0.50) GRM5SORT1SMN1; SMN2SMARCA2SMARCA4
SCHEMBL1797572 0.80 GRM5 (0.51) GRM5SORT1SMARCA2SMARCA4MEN1
SCHEMBL1797599 0.79 ABL1 (0.53) GRM5SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL1794680 0.79 GRM5 (0.55) GRM5SORT1SMN1; SMN2SMARCA2SMARCA4
SCHEMBL1798486 0.78 SMN1; SMN2 (0.47) GRM5SMN1; SMN2MEN1KMT2AKMO
SCHEMBL1797438 0.78 GRM5 (0.57) GRM5ATR
SCHEMBL4769554 0.78 KMO (0.50) SMN1; SMN2KMOMAPTNPC1RAB9A
SCHEMBL1794247 0.75 SORT1 (0.54) GRM5SORT1SMARCA2SMARCA4MEN1
SCHEMBL1796391 0.74 SMARCA2 (0.48) GRM5SORT1SMN1; SMN2SMARCA2SMARCA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed