SCHEMBL17952989

SCHEMBL17952989

CC1=Cc2c(cccc2N2CCCc3ccccc32)C1CC1C(C)=Cc2c1cccc2N1c2ccccc2CCC1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 6/20 0.35
CHRM4 P08173 6/20 0.35
CHRM1 P11229 6/20 0.35
CHRM3 P20309 5/20 0.35
CYP2D6 P10635 1/20 0.33
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
OPRL1 P41146 1/20 0.32
JAK2 O60674 1/20 0.31
JAK3 P52333 1/20 0.31
PTK2 Q05397 1/20 0.31
HTR1A P08908 2/20 0.31
ROCK1 Q13464 1/20 0.31
NUDT1 P36639 1/20 0.31
RXRA P19793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17952996 0.94 CHRM2 (0.34) CHRM2CHRM4CHRM1CHRM3POLB
SCHEMBL17952988 0.92 ROCK1 (0.34) CHRM2CHRM4CHRM1CHRM3CYP2D6
SCHEMBL17169026 0.91 L3MBTL1 (0.37) CHRM2CHRM4CHRM1CHRM3POLB
SCHEMBL17169025 0.89 MEN1 (0.38) L3MBTL1MEN1ALDH1A1KMT2AJAK2
SCHEMBL17952987 0.87 JAK2 (0.38) L3MBTL1MEN1ALDH1A1KMT2AJAK2
SCHEMBL17952991 0.86 ROCK1 (0.35) CHRM2CHRM4CHRM1CHRM3POLB
SCHEMBL19336703 0.86 CHRM2 (0.33) CHRM2CHRM4CHRM1CHRM3CYP2D6
SCHEMBL17952995 0.86 ROCK1 (0.35) CHRM2CHRM4CHRM1CHRM3POLB
SCHEMBL17952986 0.83 RXRA (0.33) CHRM2CHRM4CHRM1CHRM3POLB
SCHEMBL17169024 0.83 SMN1; SMN2 (0.39) MEN1ALDH1A1KMT2AROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9790240-B2 Ligand compound, a preparation method thereof, a transition metal compound, and a preparation method thereof LG CHEM, LTD. (KR) 2017-10-17 US disclosed
US-20160215004-A1 A NOVEL LIGAND COMPOUND, A PREPARATION METHOD THEREOF, A TRANSITION METAL COMPOUND, AND A PREPARATION METHOD THEREOF LG CHEM, LTD. (KR) 2016-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160215004-A1 A NOVEL LIGAND COMPOUND, A PREPARATION METHOD THEREOF, A TRANSITION METAL COMPOUND, AND A PREPARATION METHOD THEREOF CD40LG, OSTC, TNFSF10 CHRM2 2987/4885CHRM4 1369/4885CHRM1 2666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.