SCHEMBL17974229

SCHEMBL17974229

Nc1cccc(Nc2nccc3cc(Cl)ccc23)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.46
MAP4K4 O95819 1/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
ROCK1 Q13464 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
TNF P01375 2/20 0.43
FADS1 O60427 1/20 0.39
NR4A2 P43354 2/20 0.38
SOS2 Q07890 1/20 0.38
EGFR P00533 4/20 0.38
SCN5A Q14524 2/20 0.38
MAT2A P31153 1/20 0.37
ERBB3 P21860 1/20 0.37
JAK2 O60674 2/20 0.37
TYK2 P29597 2/20 0.37
ASIC3 Q9UHC3 1/20 0.36
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17963935 0.89 SCN9A (0.46) SCN9AMAP4K4HTR3EHTR3BHTR3A
SCHEMBL17974329 0.81 TNF (0.40) SCN9AMAP4K4HTR3EHTR3BHTR3A
SCHEMBL17963889 0.80 SCN9A (0.42) SCN9AHTR3EHTR3BHTR3AROCK1
SCHEMBL31240734 0.80 HTR3E (0.50) SCN9AHTR3EHTR3BHTR3AROCK1
SCHEMBL17974207 0.78 SCN9A (0.40) SCN9AHTR3EHTR3BHTR3AROCK1
SCHEMBL17974228 0.78 JAK2 (0.43) SCN9AHTR3EHTR3BHTR3AROCK1
SCHEMBL17974227 0.76 ASIC3 (0.42) ASIC3
SCHEMBL17963969 0.73 HSD11B1 (0.42) SCN9ASCN5AJAK2TYK2ASIC3
SCHEMBL17974204 0.73 ROCK1 (0.47) SCN9AROCK1TNFEGFRASIC3
SCHEMBL30824385 0.72 TNF (0.51) TNFFADS1EGFRSCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016120808-A1 HETEROARYLAMINOISOQUINOLINES, METHODS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF MINORYX THERAPEUTICS S.L. (ES) 2016-08-04 WO disclosed