SCHEMBL17993474

SCHEMBL17993474

Cc1ccc(-c2ccc3oc4ccc(-n5c6ccccc6n6c7ccccc7nc56)cc4c3c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.38
POLB P06746 3/20 0.38
FLT3 P36888 2/20 0.37
ALDH1A1 P00352 7/20 0.35
KDM4E B2RXH2 5/20 0.35
PIK3CD O00329 2/20 0.35
PIK3CA P42336 2/20 0.35
SMN1; SMN2 Q16637 5/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HSD17B10 Q99714 2/20 0.35
TP53 P04637 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
GAA P10253 3/20 0.34
LMNA P02545 2/20 0.34
LCK P06239 1/20 0.34
SRC P12931 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19731968 0.94 GABRP (0.35) HPGDPOLBFLT3ALDH1A1KDM4E
SCHEMBL12800969 0.93 CHEK2 (0.33) HPGDPOLBALDH1A1KDM4ESMN1; SMN2
SCHEMBL17993513 0.92 TP53 (0.38) HPGDPOLBFLT3KDM4ESMN1; SMN2
SCHEMBL12800986 0.91 GABRP (0.37) HPGDPOLBALDH1A1KDM4ESMN1; SMN2
SCHEMBL19521865 0.91 KDM4E (0.36) HPGDPOLBFLT3ALDH1A1KDM4E
SCHEMBL21412960 0.90 HPGD (0.34) HPGDPOLBFLT3ALDH1A1KDM4E
SCHEMBL16388451 0.90 ALDH1A1 (0.33) HPGDFLT3ALDH1A1KDM4ESMN1; SMN2
SCHEMBL19275393 0.90 PDE10A (0.36) HPGDPOLBKDM4ESMN1; SMN2NPC1
SCHEMBL12800973 0.89 ADORA2B (0.33) HPGDALDH1A1KDM4EPIK3CDPIK3CA
SCHEMBL12800967 0.89 CHEK2 (0.33) HPGDPOLBALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054498-B1 BISIMIDAZODIAZOCINES IDEMITSU KOSAN CO (JP) 2017-09-20 EP disclosed
WO-2016125110-A1 BISIMIDAZOLODIAZOCINES IDEMITSU KOSAN CO., LTD. (JP) 2016-08-11 WO disclosed
EP-3054498-A1 Bisimidazodiazocines Idemitsu Kosan Co., Ltd. (JP) 2016-08-10 EP disclosed