SCHEMBL1800645

SCHEMBL1800645

CCNc1ccc(C)c(F)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.50
ALDH1A1 P00352 4/20 0.50
MEN1 O00255 3/20 0.50
MAPT P10636 3/20 0.50
HTR2C P28335 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.42
HTT P42858 1/20 0.42
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
DHODH Q02127 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6738468 0.83 ALDH1A1 (0.42) KMT2AALDH1A1MEN1MAPTSMN1; SMN2
SCHEMBL29659123 0.83 MAPT (0.46) KMT2AALDH1A1MEN1MAPTSMN1; SMN2
SCHEMBL631579 0.83 MAPT (0.46) KMT2AALDH1A1MEN1MAPTSMN1; SMN2
SCHEMBL26325050 0.82 ALDH1A1 (0.50) KMT2AALDH1A1MEN1MAPTHTR2C
SCHEMBL15757174 0.82 MAPT (0.49) KMT2AALDH1A1MEN1MAPTHTR2C
SCHEMBL30536438 0.80 ALDH1A1 (0.55) KMT2AALDH1A1MEN1MAPTSMN1; SMN2
SCHEMBL1803111 0.80 ALDH1A1 (0.55) KMT2AALDH1A1MEN1MAPTSMN1; SMN2
SCHEMBL21872428 0.79 KMT2A (0.47) KMT2AALDH1A1MEN1MAPTHTR2C
SCHEMBL17048383 0.78 MAPT (0.40) KMT2AALDH1A1MEN1MAPTTSHR
SCHEMBL8292658 0.78 ABL1 (0.40) KMT2AALDH1A1MEN1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230303570-A1 KINASE INHIBITORS AND USES THEREOF ABM THERAPEUTICS CORP (US) 2023-09-28 US disclosed
WO-2021219828-A1 NEW IMIDAZOLONE DERIVATIVES AS INHIBITORS OF PROTEIN KINASES IN PARTICULAR DYRK1A, CLK1 AND/OR CLK4 PERHA PHARMACEUTICALS (FR) 2021-11-04 WO disclosed
US-10689331-B2 IDO inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2020-06-23 US disclosed
US-20190002402-A1 IDO INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2019-01-03 US disclosed
US-8304406-B2 Compounds for treating pulmonary hypertension BAYER INTELLECTUAL PROPERTY GMBH (DE) 2012-11-06 US disclosed
US-8278455-B2 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication JANSSEN PHARMACEUTICA N.V. (BE) 2012-10-02 US disclosed
US-8278455-B2 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication JANSSEN PHARMACEUTICA N.V. (BE) 2012-10-02 US disclosed
US-20110263597-A1 SUBSTITUTED PYRIDINES AND PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY BAYER HEALTHCARE LLC (US) 2011-10-27 US disclosed
US-7977333-B2 Hyperpermeability; diabetic retinopathy, ischemic retinal-vein occlusion, prematurity, age-related macular degeneration BAYER HEALTHCARE LLC (US) 2011-07-12 US disclosed
US-7951950-B2 PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARMACEUTICALS, INC. (US) 2011-05-31 US disclosed
US-20090062278-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION JANSSEN SCIENCES IRELAND UC (IE) 2009-03-05 US disclosed
CN-101146776-A PGD2 receptor antagonists for the treatment of inflammatory diseases MILLENNIUM PHARM INC (US) 2008-03-19 CN disclosed
EP-1861372-A1 PGD2 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-12-05 EP disclosed
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication BONFANTI JEAN-FRANCOIS 2007-04-26 US disclosed
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication BONFANTI JEAN-FRANCOIS 2007-04-26 US disclosed
US-20060241109-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-10-26 US disclosed
WO-2006091674-A1 PGD2 RECEPTOR ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES MILLENNIUM PHARMACEUTICALS, INC. (US) 2006-08-31 WO disclosed
US-20040082661-A1 Urea derivatives having vanilloid receptor (vr1) antagonist activity SMITHKLINE BEECHAM P.L.C. (GB) 2004-04-29 US disclosed
EP-1366020-A1 UREA DERIVATIVES HAVING VANILLOID RECEPTOR (VR1) ANTAGONIST ACTIVITY SMITHKLINE BEECHAM PLC (GB) 2003-12-03 EP disclosed
WO-2002072536-A1 UREA DERIVATIVES HAVING VANILLOID RECEPTOR (VR1) ANTAGONIST ACTIVITY SMITHKLINE BEECHAM P.L.C. (GB) 2002-09-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230303570-A1 KINASE INHIBITORS AND USES THEREOF ERBB2, ERBB3, ERBB4 KMT2A 1095/4885ALDH1A1 1859/4885MEN1 1392/4885
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, SUB1, HYOU1 KMT2A 869/4885ALDH1A1 3108/4885MEN1 2273/4885
US-20090062278-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CYC1, SUB1 KMT2A 835/4885ALDH1A1 2167/4885MEN1 2129/4885
US-20110263597-A1 SUBSTITUTED PYRIDINES AND PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY VEGFA, PGF, FLT1 KMT2A 3738/4885ALDH1A1 1173/4885MEN1 3778/4885
US-20190002402-A1 IDO INHIBITORS IDO1, IDO2, INMT KMT2A 461/4885ALDH1A1 707/4885MEN1 2981/4885
US-20040082661-A1 Urea derivatives having vanilloid receptor (vr1) antagonist activity UTS2R, TRPV1, VRK1 KMT2A 4125/4885ALDH1A1 1337/4885MEN1 4379/4885
US-10689331-B2 IDO inhibitors IDO1, IDO2, INMT KMT2A 461/4885ALDH1A1 707/4885MEN1 2981/4885
US-20060241109-A1 PGD2 receptor antagonists for the treatment of inflammatory diseases PTGER2, PTGDR2, PTGER1 KMT2A 4505/4885ALDH1A1 2836/4885MEN1 4590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.