SCHEMBL18007656

SCHEMBL18007656

NS(=O)(=O)c1cnc2c(c1)CCC2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 8/20 0.53
CA2 P00918 8/20 0.53
CA12 O43570 4/20 0.53
CA7 P43166 2/20 0.53
CA14 Q9ULX7 2/20 0.53
CCNT1 O60563 1/20 0.43
CDK1 P06493 1/20 0.43
CCNB1 P14635 1/20 0.43
CCNA2 P20248 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CCND3 P30281 1/20 0.43
FLT3 P36888 1/20 0.43
CDK9 P50750 1/20 0.43
CDK6 Q00534 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43
CA9 Q16790 4/20 0.41
ADRA2A P08913 3/20 0.41
ADRA2B P18089 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31135860 1.00 CA1 (0.53) CA1CA2CA12CA7CA14
SCHEMBL28304436 0.96 CA1 (0.49) CA1CA2CA12CA7CA14
SCHEMBL29650253 0.79 ADRA2A (0.41) CA1CA2CA12CA7CA14
SCHEMBL19693184 0.79 ADRA2A (0.41) CA1CA2CA12CA7CA14
Hydrochloric Acid SCHEMBL28291820 0.77 ADRA2A (0.47) CA1CA2CA12CA7CA14
SCHEMBL21327723 0.73 CHRNA7 (0.54)
SCHEMBL5464319 0.71 ADRA2A (0.47) ADRA2AADRA2BADRA2CLMNACYP11B2
SCHEMBL29791251 0.71 ADRA2A (0.47) ADRA2AADRA2BADRA2CLMNACYP11B2
SCHEMBL29519756 0.69 CA1 (1.00) CA1CA2CA12CA7CA14
SCHEMBL2011443 0.69 CA1 (1.00) CA1CA2CA12CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240400502-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME UNIV QUEENSLAND (AU) 2024-12-05 US disclosed
US-11845715-B2 2023-12-19 US disclosed
US-20220112159-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME UNIV QUEENSLAND (AU) 2022-04-14 US disclosed
EP-3888749-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME The University of Queensland (AU) 2021-10-06 EP disclosed
US-11130731-B2 Sulfonylureas and related compounds and use of same THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2021-09-28 US disclosed
EP-3578547-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME The University of Queensland (AU) 2019-12-11 EP disclosed
US-20180044287-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME INFLAZOME LIMITED (IE) 2018-02-15 US disclosed
EP-3259253-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME The University of Queensland (AU) 2017-12-27 EP disclosed
WO-2016131098-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME THE UNIVERSITY OF QUEENSLAND (AU) 2016-08-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220112159-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME NLRP3, PYCARD, IAPP CA1 4141/4885CA2 2434/4885CA12 4653/4885
US-11845715-B2 NLRP3, PYCARD, NOD1 CA1 4541/4885CA2 3818/4885CA12 4772/4885
US-11130731-B2 Sulfonylureas and related compounds and use of same NLRP3, PYCARD, IAPP CA1 4141/4885CA2 2434/4885CA12 4653/4885
US-20240400502-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME NLRP3, PYCARD, IAPP CA1 4141/4885CA2 2434/4885CA12 4653/4885
US-20180044287-A1 SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME NLRP3, PYCARD, IAPP CA1 4141/4885CA2 2434/4885CA12 4653/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.