SCHEMBL18017455

SCHEMBL18017455

COC(=O)c1cncc(CN(C)C(=O)c2ccc(C[C@@H]3CC[C@H]([C@H](O[SiH](C)C(C)(C)C)c4ccccc4)N3C(=O)OC(C)(C)C)cc2)c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CETP P11597 4/20 0.34
LIMK2 P53671 1/20 0.32
ABL1 P00519 1/20 0.32
RIN1 Q13671 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
SLC2A1 P11166 1/20 0.31
GPR119 Q8TDV5 2/20 0.31
CCR5 P51681 1/20 0.31
JAK2 O60674 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
USP30 Q70CQ3 1/20 0.30
ACKR3 P25106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18017454 0.90 CETP (0.35) CETPLIMK2ABL1RIN1SLC2A1
SCHEMBL16630680 0.90 CETP (0.34) CETPLIMK2ABL1RIN1HDAC1
SCHEMBL16629823 0.89 CETP (0.36) CETPLIMK2ABL1RIN1HDAC1
SCHEMBL17986551 0.83 LIMK2 (0.33) CETPLIMK2ABL1RIN1SLC2A1
SCHEMBL16629922 0.83 P2RX3 (0.34) HDAC1HDAC6GPR119
SCHEMBL18210813 0.81 CYP3A4 (0.33) CETPSLC2A1GPR119
SCHEMBL16629854 0.80 P2RX3 (0.31) CETPGPR119
SCHEMBL16619381 0.80 CETP (0.36) CETPLIMK2ABL1RIN1HDAC1
SCHEMBL16629857 0.80 CETP (0.36) CETPLIMK2ABL1RIN1HDAC1
SCHEMBL18017460 0.80 CETP (0.34) CETPLIMK2ABL1RIN1GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160235727-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2016-08-18 US disclosed
US-20160235727-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2016-08-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160235727-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS ADRB3, ADRB1, ADRB2 CETP 3055/4885LIMK2 3471/4885ABL1 3286/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.