SCHEMBL1809309

SCHEMBL1809309

COC(=O)c1sc2cnc(Cl)cc2c1CBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.40
ALDH1A1 P00352 5/20 0.40
HPGD P15428 5/20 0.40
GAA P10253 4/20 0.40
GLA P06280 3/20 0.40
HSD17B10 Q99714 3/20 0.40
CASP1 P29466 1/20 0.40
HTT P42858 1/20 0.40
CASP7 P55210 1/20 0.40
NCOA1 Q15788 1/20 0.40
RCE1 Q9Y256 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
KMT2A Q03164 5/20 0.36
NPSR1 Q6W5P4 2/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1808127 0.81 HPGD (0.44) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL7834912 0.80 KDM4E (0.59) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1808276 0.78 GABRP (0.45) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1809198 0.77 GABRA1 (0.48) KDM4EALDH1A1HPGDGAAHSD17B10
SCHEMBL31564753 0.76 L3MBTL1 (0.49) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1269967 0.72 LMNA (0.63) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1808049 0.72 GABRP (0.40) KDM4EALDH1A1HPGDGAAHTT
SCHEMBL25235837 0.72 KDM4E (0.56) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1808140 0.72 KMT2A (0.41) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL1810544 0.68 KMT2A (0.59) KDM4EALDH1A1HPGDGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011056725-A1 PYRIDINE DERIVATIVES AND METHODS OF USE THEREOF CRYSTALGENOMICS, INC. (KR) 2011-05-12 WO disclosed