SCHEMBL18106910

SCHEMBL18106910

Nc1cccc2[nH]c(NC(=O)O)nc12.c1ccc(C2CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.45
ADORA2A P29274 3/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
SMN1; SMN2 Q16637 5/20 0.42
CHEK1 O14757 1/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 5/20 0.41
POLB P06746 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 1/20 0.40
LPAR2 Q9HBW0 1/20 0.40
CYP3A4 P08684 1/20 0.40
HTR2B P41595 1/20 0.39
PARP1 P09874 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
LIPG Q9Y5X9 1/20 0.39
IDO1 P14902 1/20 0.39
PKM P14618 1/20 0.39
RIPK1 Q13546 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18106906 0.82 SMN1; SMN2 (0.63) MAOBADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL18106900 0.81 SMN1; SMN2 (0.48) MAOBADORA2AADORA2BADORA1SMN1; SMN2
SCHEMBL15944991 0.80 LPAR2 (0.59) MAOBADORA2AADORA2BADORA1SMN1; SMN2
SCHEMBL6118295 0.78 MAOB (0.71) MAOBADORA2AADORA2BADORA1SMN1; SMN2
SCHEMBL1012546 0.76 LMNA (0.59) MAOBADORA2AADORA2BADORA1SMN1; SMN2
SCHEMBL18106893 0.76 TUBB4A (0.51) SMN1; SMN2NPC1RAB9APOLBTDP1
SCHEMBL18106895 0.75 LPAR2 (0.67) MAOBADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL18106907 0.75 NPC1 (0.60) MAOBADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL18106909 0.74 RAB9A (0.60) MAOBADORA2ASMN1; SMN2NPC1RAB9A
SCHEMBL18106896 0.74 NPC1 (0.60) MAOBADORA2ASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2742029-B1 N-(BENZIMIMDAZOL-2-YL)-CYCLOPROPANE CARBOXAMIDES AS LYSOPHOSPHATIDIC ACID ANTAGONISTS MERCK PATENT GMBH (DE) 2016-10-05 EP claimed