SCHEMBL18113975

SCHEMBL18113975

C#Cc1nc2c([nH]1)c(=O)[nH]c(=O)n2Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.56
TLR7 Q9NYK1 4/20 0.50
ADORA3 P0DMS8 5/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
KDM4E B2RXH2 3/20 0.49
HPGD P15428 3/20 0.49
TSHR P16473 2/20 0.49
PSMD14 O00487 1/20 0.49
HTT P42858 1/20 0.49
ALDH1A1 P00352 2/20 0.47
BRD4 O60885 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
HSD17B10 Q99714 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
MCL1 Q07820 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4624542 0.80 PNP (0.60) PNPTLR7ADORA3MEN1KMT2A
SCHEMBL5641835 0.80 PNP (0.60) PNPTLR7ADORA3MEN1KMT2A
SCHEMBL18113976 0.79 ADORA2B (0.48) ADORA3MEN1KMT2AKDM4EHPGD
SCHEMBL22560010 0.77 PNP (0.65) PNPTLR7HPGDALDH1A1ADORA2A
SCHEMBL4202515 0.76 PNP (0.53) PNPTLR7ADORA3MEN1KMT2A
SCHEMBL4193079 0.75 PNP (0.52) PNPTLR7ADORA3MEN1KMT2A
SCHEMBL8355232 0.73 ADORA3 (0.65) PNPTLR7ADORA3MEN1KMT2A
SCHEMBL9032111 0.72 PNP (1.00) PNPTLR7ADORA3KMT2AHPGD
SCHEMBL9904017 0.71 GAA (0.47) KMT2AKDM4EHPGDTSHRALDH1A1
SCHEMBL1948025 0.71 ADORA2B (0.67) ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016159746-A1 NOVEL ETHYNYLXANTHINES, THEIR PREPARATION AND USE AS INHIBITORS OF MATRIX METALLOPROTEINASES AND ANGIOGENESIS LATVIAN INSTITUTE OF ORGANIC SYNTHESIS (LV) 2016-10-06 WO disclosed