SCHEMBL8355232

SCHEMBL8355232

O=c1[nH]c(=O)n(Cc2ccccc2)c2nc(C3CCCC3)[nH]c12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.65
ADORA1 P30542 6/20 0.65
ADORA2A P29274 5/20 0.63
ADORA2B P29275 4/20 0.63
KMT2A Q03164 5/20 0.59
PNP P00491 1/20 0.53
MEN1 O00255 4/20 0.47
POLB P06746 1/20 0.47
RAB9A P51151 1/20 0.47
TSHR P16473 2/20 0.47
GMNN O75496 1/20 0.47
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
PMP22 Q01453 1/20 0.47
HIF1A Q16665 1/20 0.47
TLR7 Q9NYK1 1/20 0.47
KDM4E B2RXH2 1/20 0.46
PSMD14 O00487 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8576753 0.87 ADORA1 (0.60) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8575318 0.81 ADORA1 (0.65) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL5229239 0.80 ADORA3 (0.61) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8358871 0.80 ADORA3 (0.94) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL9170264 0.79 ADORA1 (0.62) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8355407 0.79 ADORA3 (1.00) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8118476 0.79 ADORA1 (1.00) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8020381 0.78 ADORA2B (0.68) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL8579784 0.78 ADORA1 (0.65) ADORA3ADORA1ADORA2AADORA2BKMT2A
SCHEMBL5229734 0.78 ADORA2B (1.00) ADORA3ADORA1ADORA2AADORA2BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031101-A1 ADENOSINE RECEPTOR ANTAGONISTS WITH IMPROVED BIOACTIVITY UNIVERSITY OF SOUTH FLORIDA (US) 1999-06-24 WO disclosed