SCHEMBL1811490

SCHEMBL1811490

Clc1ccc(C2CCC(c3onc4c3CCc3c[c]ccc3-4)CC2)cc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.34
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
TSHR P16473 1/20 0.30
DRD4 P21917 1/20 0.30
DRD3 P35462 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1807788 0.77 S1PR1 (0.45) GPBAR1CYP3A4
SCHEMBL1808235 0.77 GPBAR1 (0.32) GPBAR1
SCHEMBL1813449 0.70 S1PR1 (0.54) CYP3A4
SCHEMBL315186 0.62 HTR3A (0.58) MEN1CYP1A2TSHRKMT2A
SCHEMBL134194 0.60
SCHEMBL482279 0.58 HTR3A (0.48) MEN1CYP1A2TSHRKMT2A
SCHEMBL18533598 0.57 HTR3A (0.52) MEN1CYP1A2TSHRKMT2A
Methyl Alcohol SCHEMBL15391253 0.57 DRD2 (0.55) MEN1CYP1A2TSHRKMT2A
SCHEMBL28101829 0.57 SLC18A3 (0.40) MEN1KMT2A
SCHEMBL22929 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011059784-A1 TRICYCLIC HETEROCYCLIC COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed