SCHEMBL18153773

SCHEMBL18153773

COc1ccc(CN(O)C(=O)c2ccc3c(c2)CCC2(CCNC2)C3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ACHE P22303 1/20 0.36
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
HTR2A P28223 1/20 0.35
PDK1 Q15118 3/20 0.34
PDK2 Q15119 3/20 0.34
PDK3 Q15120 3/20 0.34
PDK4 Q16654 3/20 0.34
ADRA2A P08913 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ABCB1 P08183 1/20 0.33
ABCC1 P33527 1/20 0.33
CTSS P25774 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18152170 0.96 MEN1 (0.39) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18153740 0.91 ALOX5 (0.41) MEN1KMT2AOPRM1OPRD1ADRA2A
SCHEMBL18152111 0.86 HSD17B2 (0.40) MEN1KMT2AOPRM1OPRD1NPC1
SCHEMBL18152144 0.83 OPRM1 (0.38) OPRM1OPRD1ADRA2ANPC1RAB9A
SCHEMBL18153894 0.80 MEN1 (0.38) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18153708 0.80 MEN1 (0.38) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18152186 0.80 CYP2D6 (0.38) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18152041 0.78 MEN1 (0.39) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18152127 0.77 MEN1 (0.38) MEN1KMT2AACHEOPRM1OPRD1
SCHEMBL18152169 0.77 MEN1 (0.38) MEN1KMT2AACHEOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016168660-A1 3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-20 WO disclosed