SCHEMBL18153791

SCHEMBL18153791

COc1ccc(C(=O)N(O)C(=O)c2ccc3c(c2)CCC2(CCNCC2)O3)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.44
HTR2C P28335 3/20 0.44
DRD2 P14416 2/20 0.44
OPRD1 P41143 6/20 0.41
OPRM1 P35372 4/20 0.41
HRH3 Q9Y5N1 2/20 0.39
RXRA P19793 1/20 0.38
KCNH2 Q12809 4/20 0.37
CYP2D6 P10635 3/20 0.37
GPR183 P32249 1/20 0.37
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
OPRL1 P41146 1/20 0.35
ALDH1A1 P00352 1/20 0.35
F2 P00734 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18152038 0.92 OPRD1 (0.41) HTR2AHTR2CDRD2OPRD1OPRM1
SCHEMBL18144919 0.79 OPRD1 (0.45) HTR2AHTR2CDRD2OPRD1HRH3
Hydrochloric Acid SCHEMBL8567312 0.79 HTR2A (0.56) HTR2AHTR2CDRD2OPRD1HRH3
SCHEMBL18152041 0.79 MEN1 (0.39) HTR2AHTR2CDRD2OPRD1OPRM1
SCHEMBL18165461 0.78 RXRA (0.43) HTR2AHTR2CDRD2OPRD1HRH3
SCHEMBL18152144 0.76 OPRM1 (0.38) OPRD1OPRM1KCNH2KDM4EHPGD
SCHEMBL28524517 0.72 HTR2C (0.52) HTR2AHTR2CDRD2OPRD1OPRM1
SCHEMBL18148508 0.70 OPRD1 (0.45) OPRD1RXRAKCNH2ALDH1A1KMT2A
SCHEMBL11254881 0.70 HTR2C (0.49) HTR2AHTR2CDRD2OPRD1HRH3
SCHEMBL18144845 0.69 HDAC6 (0.55) HTR2AHTR2CDRD2CYP2D6GPR183

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016168660-A1 3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-20 WO claimed
WO-2016168660-A1 3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-20 WO disclosed