SCHEMBL1815423

SCHEMBL1815423

Cc1ccc(OCC(=O)NC(c2ccccc2)c2cc(Cl)c3cccnc3c2O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 19/20 1.00
ADAMTS4 O75173 2/20 0.74
KDM4E B2RXH2 1/20 0.73
ALOX12 P18054 1/20 0.73
L3MBTL1 Q9Y468 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1812589 0.96 ADAMTS5 (1.00) ADAMTS5ADAMTS4KDM4EALOX12L3MBTL1
SCHEMBL1814568 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4
SCHEMBL3976904 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4
SCHEMBL1812659 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4
SCHEMBL1815616 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4
SCHEMBL1812131 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4KDM4EALOX12L3MBTL1
SCHEMBL1816647 0.93 ADAMTS5 (0.95) ADAMTS5ADAMTS4
SCHEMBL1812713 0.93 ADAMTS5 (1.00) ADAMTS5ADAMTS4
SCHEMBL1817552 0.93 ADAMTS5 (0.86) ADAMTS5ADAMTS4KDM4EALOX12
SCHEMBL1814842 0.92 ADAMTS5 (0.89) ADAMTS5ADAMTS4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101505751-A 8-hydroxyquinoline compounds and methods thereof WYETH CORP (US) 2009-08-12 CN claimed
EP-2056823-A2 8-HYDROXYQUINOLINE COMPOUNDS AND METHODS THEREOF Wyeth (US) 2009-05-13 EP claimed
US-20080269213-A1 8-Hydroxyquinoline compounds and methods thereof WYETH (US) 2008-10-30 US claimed
WO-2008024922-A2 8-HYDROXYQUINOLINE COMPOUNDS AND METHODS THEREOF WYETH (US) 2008-02-28 WO claimed
US-7947712-B2 Antiarthritic agents; asthma; chronic obstructive pulminary diosrders; atherosclerosis; vision defects; hepatitis; central nervous system disorders; cardiovascular disorders; wound healing agents; restenosis; cirrhosis; multiple sclerosis; glomerulonephritis; graft versus host disease; antidiabetic agent WYETH LLC (US) 2011-05-24 US disclosed
CN-101505751-A 8-hydroxyquinoline compounds and methods thereof WYETH CORP (US) 2009-08-12 CN disclosed
EP-2056823-A2 8-HYDROXYQUINOLINE COMPOUNDS AND METHODS THEREOF Wyeth (US) 2009-05-13 EP disclosed
US-20080269213-A1 8-Hydroxyquinoline compounds and methods thereof WYETH (US) 2008-10-30 US disclosed
WO-2008024922-A2 8-HYDROXYQUINOLINE COMPOUNDS AND METHODS THEREOF WYETH (US) 2008-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269213-A1 8-Hydroxyquinoline compounds and methods thereof MMP8, MMP26, MMP9 ADAMTS5 11/4885ADAMTS4 14/4885KDM4E 4164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.