SCHEMBL1816201

SCHEMBL1816201

NC(=O)c1ccc(N2CC(C(=O)O)C2)cc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 18/20 0.56
S1PR1 P21453 1/20 0.45
S1PR3 Q99500 1/20 0.45
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1817248 0.87 NOTUM (0.60) NOTUMS1PR1PDK2
SCHEMBL3598011 0.76 ABHD6 (0.46) NOTUM
SCHEMBL15547228 0.73 WDR5 (0.44) NOTUM
SCHEMBL2968971 0.72 NOTUM (0.65) NOTUM
SCHEMBL2431606 0.71 HRH3 (0.52)
SCHEMBL24177167 0.71 CES2 (0.47)
SCHEMBL29789661 0.71 CES2 (0.47)
SCHEMBL15923406 0.71 IP6K1 (0.58) NOTUM
Trifluoroacetic Acid SCHEMBL3475248 0.71 HRH3 (0.49)
SCHEMBL2938165 0.69 NOTUM (0.75) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951805-B2 Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase XENON PHARMACEUTICALS INC. (CA) 2011-05-31 US disclosed