SCHEMBL18166300

SCHEMBL18166300

CCOCc1nnnn1-c1cc(OC(=O)NC(C)c2nccs2)cc(-c2ccc(C)cc2)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.46
P2RX2 Q9UBL9 1/20 0.46
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 4/20 0.33
MAPT P10636 2/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
CTSA P10619 3/20 0.32
MEN1 O00255 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2C19 P33261 2/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166451 0.92 P2RX3 (0.45) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL18166450 0.92 P2RX3 (0.54) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL18166339 0.91 P2RX3 (0.48) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL10243504 0.88 P2RX3 (0.60) P2RX3P2RX2NPC1RAB9ALMNA
SCHEMBL18166362 0.86 P2RX3 (0.41) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL18166330 0.85 P2RX3 (0.65) P2RX3P2RX2
SCHEMBL18036366 0.84 P2RX3 (0.45) P2RX3P2RX2GAALMNAMAPT
SCHEMBL18166396 0.83 P2RX3 (0.39) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL18166418 0.83 P2RX3 (0.39) P2RX3P2RX2NPC1RAB9AGAA
SCHEMBL18036358 0.82 P2RX3 (0.44) P2RX3P2RX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed