SCHEMBL18166384

SCHEMBL18166384

Cc1ccc(-c2cc(OC(=O)NCc3cccc(C)n3)cc(-n3nnnc3C(C)C)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.36
P2RX2 Q9UBL9 2/20 0.36
IRAK4 Q9NWZ3 1/20 0.34
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
EPHX1 P07099 1/20 0.33
MAP3K5 Q99683 2/20 0.33
ALOX5 P09917 1/20 0.33
PTGS1 P23219 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166295 0.92 P2RX3 (0.35) P2RX3P2RX2EPHX1MAP3K5ALOX5
SCHEMBL18166448 0.92 P2RX3 (0.35) P2RX3P2RX2ALDH1A1TSHREPHX1
SCHEMBL18166446 0.86 P2RX3 (0.45) P2RX3P2RX2
SCHEMBL10244122 0.86 P2RX3 (0.45) P2RX3P2RX2IRAK4TSHR
SCHEMBL18166368 0.84 P2RX3 (0.47) P2RX3P2RX2EPHX1
SCHEMBL18166376 0.83 P2RX3 (0.39) P2RX3P2RX2EPHX1NPC1RAB9A
SCHEMBL18166336 0.82 P2RX3 (0.40) P2RX3P2RX2
SCHEMBL18166430 0.82 ADORA2A (0.41) P2RX3P2RX2EPHX1MAP3K5
SCHEMBL18166317 0.82 P2RX3 (0.37) P2RX3P2RX2
SCHEMBL18166413 0.81 P2RX3 (0.41) P2RX3P2RX2ALDH1A1TSHREPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed