SCHEMBL18179943

SCHEMBL18179943

Cc1ccc(Br)cc1CNC12CC3CC(C)(CC(C)(C3)C1)C2

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.49
HDAC8 Q9BY41 6/20 0.49
GRIN2D O15399 2/20 0.47
GRIN3B O60391 2/20 0.47
GRIN1 Q05586 2/20 0.47
GRIN2A Q12879 2/20 0.47
GRIN2B Q13224 2/20 0.47
GRIN2C Q14957 2/20 0.47
GRIN3A Q8TCU5 2/20 0.47
HDAC1 Q13547 5/20 0.46
HDAC3 O15379 3/20 0.46
EPHX2 P34913 9/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166480 0.84 HDAC6 (0.46) HDAC6HDAC8GRIN2DGRIN3BGRIN1
SCHEMBL18170344 0.84 HDAC6 (0.46) HDAC6HDAC8GRIN2DGRIN3BGRIN1
SCHEMBL18184323 0.84 HDAC6 (0.46) HDAC6HDAC8GRIN2DGRIN3BGRIN1
SCHEMBL18170343 0.84 HDAC6 (0.46) HDAC6HDAC8GRIN2DGRIN3BGRIN1
SCHEMBL16884223 0.71 SCN9A (0.44) HDAC6HDAC8HDAC1HDAC3
SCHEMBL16884198 0.68 CNR2 (0.44) HDAC6EPHX2
SCHEMBL31137114 0.68 KDM1A (0.47) HDAC6
SCHEMBL16884338 0.68 SCN9A (0.46) HDAC6HDAC8HDAC1HDAC3
SCHEMBL22927151 0.68 CYP2D6 (0.41) HDAC6HDAC8GRIN2DGRIN3BGRIN1
SCHEMBL13641428 0.66 HDAC6 (0.45) HDAC6HDAC8HDAC1HDAC3EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10039727-B2 Adamantane or pinene derivatives for use in the treatment of chlamydiales infections COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2018-08-07 US disclosed
US-20160310448-A1 Adamantane or Pinene Derivatives for Use in the Treatment of Chlamydiales Infections COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2016-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10039727-B2 Adamantane or pinene derivatives for use in the treatment of chlamydiales infections ADRA1A, ADRA1B, ADRA1D HDAC6 4361/4885HDAC8 4222/4885GRIN2D 3507/4885
US-20160310448-A1 Adamantane or Pinene Derivatives for Use in the Treatment of Chlamydiales Infections ADRA1A, ADRA1B, ADRA1D HDAC6 4267/4885HDAC8 4223/4885GRIN2D 3513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.