SCHEMBL18170344

SCHEMBL18170344

COc1ccc(Br)cc1CNC12CC3C[C@@](C)(C1)C[C@](C)(C3)C2

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 6/20 0.46
HDAC8 Q9BY41 5/20 0.46
GRIN1 Q05586 4/20 0.43
GRIN2A Q12879 4/20 0.43
KDM1A O60341 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KDM1B Q8NB78 1/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.43
USP2 O75604 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18170343 1.00 HDAC6 (0.46) HDAC6HDAC8GRIN1GRIN2AKDM1A
SCHEMBL18184323 1.00 HDAC6 (0.46) HDAC6HDAC8GRIN1GRIN2AKDM1A
SCHEMBL18166480 1.00 HDAC6 (0.46) HDAC6HDAC8GRIN1GRIN2AKDM1A
SCHEMBL18179943 0.84 HDAC6 (0.49) HDAC6HDAC8GRIN1GRIN2AGRIN2D
SCHEMBL20959894 0.84 MEN1 (0.50) KDM1AMAOAMAOBKDM1BMEN1
SCHEMBL3359762 0.84 MEN1 (0.50) KDM1AMAOAMAOBKDM1BMEN1
Hydrochloric Acid SCHEMBL3363220 0.83 MEN1 (0.52) KDM1AMAOAMAOBKDM1BMEN1
SCHEMBL20959900 0.81 MEN1 (0.47) KDM1AMAOAMAOBKDM1BMEN1
SCHEMBL22353273 0.80 KDM1A (0.40) KDM1AMAOAMAOBKDM1BMEN1
SCHEMBL3311930 0.72 ALDH1A1 (0.38) HDAC6HDAC8GRIN1GRIN2AKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3085688-B1 ADAMANTANE OR PINENE DERIVATIVES FOR USE IN THE TREATMENT OF CHLAMYDIALES INFECTIONS COMMISSARIAT ENERGIE ATOMIQUE (FR) 2020-08-19 EP claimed
US-20160310448-A1 Adamantane or Pinene Derivatives for Use in the Treatment of Chlamydiales Infections COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2016-10-27 US claimed
EP-3085688-B1 ADAMANTANE OR PINENE DERIVATIVES FOR USE IN THE TREATMENT OF CHLAMYDIALES INFECTIONS COMMISSARIAT ENERGIE ATOMIQUE (FR) 2020-08-19 EP disclosed
US-10039727-B2 Adamantane or pinene derivatives for use in the treatment of chlamydiales infections COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2018-08-07 US disclosed
US-20160310448-A1 Adamantane or Pinene Derivatives for Use in the Treatment of Chlamydiales Infections COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2016-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10039727-B2 Adamantane or pinene derivatives for use in the treatment of chlamydiales infections ADRA1A, ADRA1B, ADRA1D HDAC6 4361/4885HDAC8 4222/4885GRIN1 1262/4885
US-20160310448-A1 Adamantane or Pinene Derivatives for Use in the Treatment of Chlamydiales Infections ADRA1A, ADRA1B, ADRA1D HDAC6 4267/4885HDAC8 4223/4885GRIN1 1157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.