SCHEMBL18198243

SCHEMBL18198243

COc1ccc(C2OCCO2)c(Br)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR2C P28335 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP4B1 P13584 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP3A5 P20815 1/20 0.36
CYP2A7 P20853 1/20 0.36
CYP3A7 P24462 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1119892 0.88 NPC1 (0.52) NPC1RAB9ACYP2C19HTR2CMAPT
SCHEMBL29404769 0.88 NPC1 (0.52) NPC1RAB9ACYP2C19HTR2CMAPT
SCHEMBL29995130 0.81 NPC1 (0.47) NPC1RAB9ACYP2C19MEN1KMT2A
SCHEMBL17796062 0.81 NPC1 (0.47) NPC1RAB9ACYP2C19MEN1KMT2A
SCHEMBL5790025 0.81 NPC1 (0.52) NPC1RAB9ACYP2C19ALDH1A1CYP1A1
SCHEMBL16682588 0.80 ALDH1A1 (0.37) NPC1RAB9AALDH1A1MAPT
SCHEMBL8493047 0.80 NAAA (0.40) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL4802700 0.79 NPC1 (0.54) NPC1RAB9ACYP2C19ALDH1A1MEN1
SCHEMBL2469533 0.77 NPC1 (0.52) NPC1RAB9ACYP2C19ALDH1A1MEN1
SCHEMBL21164867 0.77 ERN1 (0.50) NPC1RAB9ACYP2C19ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10351706-B2 Near-infrared fluorescent dyes and uses thereof EAST CHINA UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2019-07-16 US disclosed
US-20160318933-A1 FUSED PYRAZOLE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2016-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160318933-A1 FUSED PYRAZOLE DERIVATIVE DRD4, DRD2, DRD3 NPC1 3495/4885RAB9A 1241/4885CYP2C19 206/4885
US-10351706-B2 Near-infrared fluorescent dyes and uses thereof IK, CYBA, CRY2 NPC1 304/4885RAB9A 1196/4885CYP2C19 191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.