SCHEMBL18210663

SCHEMBL18210663

CC(C)Oc1cc(N2CCN(C(C)(C)C)CC2)ccc1F

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 3/20 0.39
CCR1 P32246 1/20 0.39
MAP2 P11137 2/20 0.38
NR1H2 P55055 5/20 0.36
NR1H3 Q13133 4/20 0.36
SLC6A9 P48067 1/20 0.36
DRD2 P14416 4/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
RXRA P19793 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
HTR1A P08908 3/20 0.34
HTR2A P28223 3/20 0.34
HTR7 P34969 3/20 0.34
HTR6 P50406 3/20 0.34
HIF1A Q16665 1/20 0.34
CTSK P43235 1/20 0.34
CTSC P53634 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18210772 0.84 HTR6 (0.46) PTGDRDRD2HTR1AHTR2AHTR7
SCHEMBL24625570 0.74 GAA (0.39) RXRAGRIN1GRIN2B
SCHEMBL16001188 0.70 SIRT6 (0.43) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL1709030 0.70 MAPT (0.57)
SCHEMBL11291219 0.70 ALDH1A1 (0.43) HTR7
SCHEMBL3469564 0.70 MAPK1 (0.43) CCR1HTR7
SCHEMBL19692631 0.69 AR (0.47) HTR2AHTR6CTSKCTSC
SCHEMBL16001227 0.68 SIRT6 (0.46) PTGDRHTR6
SCHEMBL21378854 0.68 HTR6 (0.50) HTR6CTSK
SCHEMBL14923962 0.67 PANK3 (0.43) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9486422-B2 Small molecule inhibitors of Mcl-1 and the uses of thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-11-08 US disclosed