SCHEMBL18210772

SCHEMBL18210772

CC(C)Oc1cc(N2CCN(C)CC2)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.46
HTR1A P08908 5/20 0.46
DRD2 P14416 5/20 0.46
HTR2A P28223 5/20 0.46
HTR7 P34969 5/20 0.46
SIRT6 Q8N6T7 1/20 0.45
HTR3A P46098 1/20 0.44
GAA P10253 3/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 2/20 0.43
PTK2B Q14289 2/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
LRRK2 Q5S007 1/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
GLA P06280 1/20 0.42
ADRA2C P18825 2/20 0.41
PTGDR Q13258 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18210663 0.84 PTGDR (0.39) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL16001227 0.83 SIRT6 (0.46) HTR6SIRT6HTR3AGAAKDM4E
SCHEMBL24783778 0.83 SIRT6 (0.58) HTR6HTR1ADRD2HTR2ASIRT6
SCHEMBL15283334 0.82 GAA (0.58) HTR6SIRT6HTR3AGAAKDM4E
SCHEMBL16001188 0.79 SIRT6 (0.43) HTR6HTR1ADRD2HTR2AHTR7
SCHEMBL25699466 0.79 MAPT (0.49) HTR6SIRT6HTR3AGAAKDM4E
SCHEMBL15283363 0.79 MAPT (0.54) HTR6SIRT6HTR3AGAAKDM4E
SCHEMBL15283343 0.77 MAPT (0.52) SIRT6HTR3AGAAKDM4EMAPT
SCHEMBL8322549 0.77 HTR3A (0.55) HTR1ADRD2SIRT6HTR3AGAA
SCHEMBL15283456 0.76 SIRT6 (0.74) HTR6SIRT6MAPTMAPK1PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9486422-B2 Small molecule inhibitors of Mcl-1 and the uses of thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-11-08 US disclosed