SCHEMBL18230478

SCHEMBL18230478

COc1ccnc(-c2nc(N)sc2C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.49
CCR5 P51681 1/20 0.49
CCR8 P51685 1/20 0.49
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
MYC P01106 1/20 0.42
WDR5 P61964 1/20 0.42
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
ADORA1 P30542 4/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 3/20 0.40
KDM4E B2RXH2 2/20 0.40
MPI P34949 1/20 0.40
PLA2G2A P14555 1/20 0.39
LMNA P02545 2/20 0.38
PLAU P00749 1/20 0.38
HPGD P15428 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19638187 0.77 ADORA1 (0.57) MYCWDR5ADORA1MAPTKDM4E
SCHEMBL30309328 0.77 ADORA1 (0.57) MYCWDR5ADORA1MAPTKDM4E
SCHEMBL17951012 0.76 MYC (0.64) MYCWDR5ADORA1ALDH1A1MAPT
SCHEMBL1850971 0.75 TGFBR1 (0.51) CCR1CCR5CCR8CYP1A2ALDH1A1
SCHEMBL30309300 0.75 TGFBR1 (0.51) CCR1CCR5CCR8CYP1A2ALDH1A1
SCHEMBL6840024 0.72 KDM4E (0.46) MYCWDR5ALDH1A1KDM4ELMNA
SCHEMBL3406257 0.72 ALDH1A1 (0.58) CCR1CCR5CCR8CYP1A2ALDH1A1
Methane SCHEMBL21386924 0.71 CCR1 (0.95) CCR1CCR5CCR8NOS3NOS1
SCHEMBL19637978 0.70 ADORA1 (0.51) MYCWDR5ADORA1ALDH1A1MAPT
SCHEMBL6839964 0.70 MYC (0.31) MYCWDR5ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016183173-A1 ANTIPARASITIC COMPOUNDS Avista Pharma Solutions (US) 2016-11-17 WO disclosed
WO-2016183173-A1 ANTIPARASITIC COMPOUNDS Avista Pharma Solutions (US) 2016-11-17 WO disclosed