SCHEMBL182445

SCHEMBL182445

O=c1[nH]c(=O)c2cc(Br)ccc2[nH]1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 2/20 0.60
CHEK1 O14757 1/20 0.60
AURKA O14965 1/20 0.60
DAPK3 O43293 1/20 0.60
PRKD3 O94806 1/20 0.60
MAP4K4 O95819 1/20 0.60
PAK4 O96013 1/20 0.60
ABL1 P00519 1/20 0.60
NTRK1 P04629 1/20 0.60
CSF1R P07333 1/20 0.60
RET P07949 1/20 0.60
MET P08581 1/20 0.60
PDGFRB P09619 1/20 0.60
PIM1 P11309 1/20 0.60
FGFR1 P11362 1/20 0.60
PDGFRA P16234 1/20 0.60
PRKACA P17612 1/20 0.60
FLT1 P17948 1/20 0.60
LTK P29376 1/20 0.60
GRK5 P34947 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17979420 0.85 CA12 (0.49) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL30013301 0.84 METAP2 (0.60) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL2730824 0.84 METAP2 (0.60) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL978028 0.82 PIM1 (0.49) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL18020128 0.81 CA12 (0.47) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL24576225 0.81 LMNA (0.50) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL1396317 0.81 CHEK1 (0.56) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL7032078 0.79 CA12 (0.40) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL615808 0.79 POLB (0.53) JAK2CHEK1AURKADAPK3PRKD3
SCHEMBL7852218 0.77 PARP1 (0.64) JAK2CHEK1AURKADAPK3PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 138 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120157623-A Biological pesticide developed based on tobacco stem vinegar, and preparation and application thereof 湖北省烟草科学研究院 2025-06-17 CN claimed
CN-119176746-B Method for preparing bisphenol A and heterocyclic compound by using waste PC 浙江大学 2025-05-30 CN claimed
CN-119176746-A Method for preparing bisphenol A and heterocyclic compound by using waste PC 浙江大学 2024-12-24 CN claimed
US-20050004117-A1 Dipeptidyl peptidase inhibitors SYRRX, INC. 2005-01-06 US claimed
US-20260092053-A1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2026-04-02 US disclosed
EP-4681774-A2 KHK INHIBITORS Gilead Sciences, Inc. (US) 2026-01-21 EP disclosed
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS GILEAD SCIENCES INC (US) 2025-11-27 US disclosed
EP-4313967-B1 KHK INHIBITORS GILEAD SCIENCES INC (US) 2025-11-12 EP disclosed
US-20250325677-A1 STAT6 DEGRADERS GILEAD SCIENCES INC (US) 2025-10-23 US disclosed
US-12410160-B2 KHK inhibitors GILEAD SCIENCES, INC. (US) 2025-09-09 US disclosed
CN-120157623-A Biological pesticide developed based on tobacco stem vinegar, and preparation and application thereof 湖北省烟草科学研究院 2025-06-17 CN disclosed
CN-120157623-A Biological pesticide developed based on tobacco stem vinegar, and preparation and application thereof 湖北省烟草科学研究院 2025-06-17 CN disclosed
WO-2004087053-A2 DIPEPTIDYL PEPTIDASE INHIBITORS SYRRX, INC. (US) 2004-10-14 WO disclosed
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO disclosed
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004117-A1 Dipeptidyl peptidase inhibitors DPP9, DPP4, DPP3 JAK2 509/4885CHEK1 3621/4885AURKA 3290/4885
US-20250325677-A1 STAT6 DEGRADERS STAT6, STAT5B, STAT1 JAK2 7/4885CHEK1 3950/4885AURKA 2905/4885
US-20260092053-A1 KHK INHIBITORS KHK, SLC5A2, HK1 JAK2 1278/4885CHEK1 2740/4885AURKA 1948/4885
US-12410160-B2 KHK inhibitors KHK, KHDRBS1, NADK JAK2 877/4885CHEK1 479/4885AURKA 141/4885
US-20250361236-A9 DIACYLGLYCEROL KINASE MODULATING COMPOUNDS DGKG, DGKB, DGKK JAK2 948/4885CHEK1 353/4885AURKA 995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.