SCHEMBL1824682

SCHEMBL1824682

COc1cc(CNCc2ccc3c(Sc4ccccc4)c(OC(N)=O)[nH]c3c2)ccc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
BCHE P06276 2/20 0.47
LMNA P02545 3/20 0.46
KMT2A Q03164 3/20 0.46
NPC1 O15118 1/20 0.46
PKM P14618 1/20 0.46
RAB9A P51151 1/20 0.46
MRGPRX1 Q96LB2 2/20 0.44
F2 P00734 1/20 0.44
F10 P00742 1/20 0.44
PRSS1 P07477 1/20 0.44
F7 P08709 1/20 0.44
HTT P42858 3/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPY1R P25929 1/20 0.43
NPY2R P49146 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1825571 0.97 ALDH1A1 (0.50) ALDH1A1BCHELMNAKMT2ANPC1
SCHEMBL1615275 0.88 TP53 (0.49) ALDH1A1BCHELMNAKMT2ANPC1
SCHEMBL1823504 0.87 TP53 (0.49) ALDH1A1KMT2ANPC1RAB9AKDM4E
SCHEMBL1826130 0.86 TP53 (0.44) ALDH1A1KMT2AKDM4EPOLBMEN1
SCHEMBL1615463 0.85 ALDH1A1 (0.52) ALDH1A1BCHELMNAKMT2AHTT
SCHEMBL1824216 0.85 TP53 (0.49) ALDH1A1KMT2ANPC1HTTKDM4E
SCHEMBL1827585 0.85 TP53 (0.53) ALDH1A1KMT2AHTTKDM4ESMN1; SMN2
SCHEMBL1822868 0.84 TP53 (0.43) ALDH1A1LMNAKMT2AKDM4ESMN1; SMN2
SCHEMBL1831867 0.84 KMT2A (0.52) KMT2ASMN1; SMN2POLBMEN1TP53
SCHEMBL1824680 0.84 MEN1 (0.54) ALDH1A1KMT2ARAB9APOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794122-B1 3-SUBSTITUTED-5- AND 6-AMINOALKYL INDOLE-2-CARBOXYLIC ACID AMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I AVENTIS PHARMA INC (US) 2011-05-04 EP claimed