SCHEMBL1825571

SCHEMBL1825571

COc1ccc(CNCc2ccc3c(Sc4ccccc4)c(OC(N)=O)[nH]c3c2)cc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
BCHE P06276 2/20 0.48
HTT P42858 3/20 0.46
LMNA P02545 3/20 0.46
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KMT2A Q03164 2/20 0.46
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
TP53 P04637 3/20 0.42
POLB P06746 1/20 0.42
NPC1 O15118 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42
SMPD1 P17405 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1824682 0.97 ALDH1A1 (0.47) ALDH1A1BCHEHTTLMNAKDM4E
SCHEMBL1615463 0.88 ALDH1A1 (0.52) ALDH1A1BCHEHTTLMNAKDM4E
SCHEMBL1823504 0.88 TP53 (0.49) ALDH1A1KDM4ESMN1; SMN2KMT2ATP53
SCHEMBL1826130 0.87 TP53 (0.44) ALDH1A1KDM4EKMT2ATP53POLB
SCHEMBL1824216 0.86 TP53 (0.49) ALDH1A1HTTKDM4ESMN1; SMN2KMT2A
SCHEMBL1827585 0.86 TP53 (0.53) ALDH1A1HTTKDM4ESMN1; SMN2KMT2A
SCHEMBL1615275 0.85 TP53 (0.49) ALDH1A1BCHELMNAKMT2ATP53
SCHEMBL1822868 0.85 TP53 (0.43) ALDH1A1LMNAKDM4ESMN1; SMN2KMT2A
SCHEMBL1831867 0.85 KMT2A (0.52) SMN1; SMN2KMT2ATP53POLBMAPT
SCHEMBL1824680 0.84 MEN1 (0.54) ALDH1A1KMT2ATP53POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794122-B1 3-SUBSTITUTED-5- AND 6-AMINOALKYL INDOLE-2-CARBOXYLIC ACID AMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I AVENTIS PHARMA INC (US) 2011-05-04 EP claimed