SCHEMBL18263262

SCHEMBL18263262

O=C(OC1C2CC3CC(C2)CC1C3)c1ccccc1NCc1cc(O)ccc1O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.47
HSP90AA1 P07900 3/20 0.46
CKS1B P61024 2/20 0.46
SKP2 Q13309 2/20 0.46
SKP1 P63208 1/20 0.46
HKDC1 Q2TB90 1/20 0.41
PTGS2 P35354 1/20 0.41
SYK P43405 1/20 0.41
RGS12 O14924 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LCK P06239 1/20 0.40
MAPT P10636 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
NOX4 Q9NPH5 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Adamantane SCHEMBL28227462 0.83 EGFR (0.55) EGFRHSP90AA1CKS1BSKP2SKP1
SCHEMBL18263261 0.81 CKS1B (0.67) EGFRHSP90AA1CKS1BSKP2SKP1
SCHEMBL182501 0.81 HSP90AA1 (0.67) EGFRHSP90AA1CKS1BSKP2SKP1
SCHEMBL6259074 0.79 EGFR (0.66) EGFRHSP90AA1HKDC1NOX4
SCHEMBL6258501 0.75 EGFR (0.63) EGFRHSP90AA1SYKRGS12ALDH1A1
SCHEMBL6260824 0.75 EGFR (0.52) EGFRHSP90AA1HKDC1SYKRGS12
SCHEMBL31060627 0.75 EGFR (0.52) EGFRHSP90AA1HKDC1SYKRGS12
SCHEMBL4973520 0.70 HSP90AA1 (0.43) EGFRHSP90AA1CKS1BSKP2SKP1
SCHEMBL17358251 0.69 HSD11B1 (0.40) ALDH1A1
SCHEMBL11510342 0.69 CA12 (0.61) EGFRHSP90AA1HKDC1SYKRGS12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016190847-A1 SUBSTITUTED HETEROARYL COMPOUNDS AND METHODS OF USE CALITOR SCIENCES, LLC (US) 2016-12-01 WO disclosed