SCHEMBL18275334

SCHEMBL18275334

CN(C(=O)c1ccc(NC(=O)Cc2ccc(S(=O)(=O)CC3CC3)cc2)cc1)C1CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 5/20 0.58
RIN1 Q13671 5/20 0.58
RORC P51449 9/20 0.56
KDM4A O75164 1/20 0.53
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ATM Q13315 1/20 0.50
HSD11B1 P28845 1/20 0.49
HSD11B2 P80365 1/20 0.49
KMT2A Q03164 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18275317 0.88 RORC (0.52) ABL1RIN1RORC
SCHEMBL18275325 0.87 RORC (0.56) RORCALDH1A1
SCHEMBL18275230 0.85 RORC (0.53) RORC
SCHEMBL18294253 0.85 RORC (0.56) RORC
SCHEMBL18275253 0.83 RORC (0.59) RORC
SCHEMBL18275323 0.83 RORC (0.62) RORC
SCHEMBL18294324 0.82 RORC (0.57) RORC
SCHEMBL18275264 0.82 RORC (0.52) ABL1RIN1RORCALDH1A1
SCHEMBL18294272 0.81 RORC (0.57) RORC
SCHEMBL18275330 0.81 RORC (0.65) ABL1RIN1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3303291-B1 ROR-GAMMA MODULATORS LEAD PHARMA B V (NL) 2020-03-18 EP claimed
US-10315996-B2 ROR gamma (RORγ) modulators LEAD PHARMA HOLDING B.V. (NL) 2019-06-11 US claimed
US-20180170877-A1 ROR GAMMA (RORY) MODULATORS LEAD PHARMA HOLDING B.V. (NL) 2018-06-21 US claimed
EP-3101006-A1 ROR GAMMA (RORY) MODULATORS Lead Pharma Cel Models IP B.V. (NL) 2016-12-07 EP claimed
CN-108473429-B ROR gamma modulators 领先制药控股公司 2021-09-10 CN disclosed
US-10315996-B2 ROR gamma (RORγ) modulators LEAD PHARMA HOLDING B.V. (NL) 2019-06-11 US disclosed
US-10315996-B2 ROR gamma (RORγ) modulators LEAD PHARMA HOLDING B.V. (NL) 2019-06-11 US disclosed
US-20180170877-A1 ROR GAMMA (RORY) MODULATORS LEAD PHARMA HOLDING B.V. (NL) 2018-06-21 US disclosed
US-20180170877-A1 ROR GAMMA (RORY) MODULATORS LEAD PHARMA HOLDING B.V. (NL) 2018-06-21 US disclosed
US-20180170877-A1 ROR GAMMA (RORY) MODULATORS LEAD PHARMA HOLDING B.V. (NL) 2018-06-21 US disclosed
WO-2016193452-A1 ROR GAMMA (RORγ) MODULATORS LEAD PHARMA CEL MODELS IP B.V. (NL) 2016-12-08 WO disclosed
EP-3101006-A1 ROR GAMMA (RORY) MODULATORS Lead Pharma Cel Models IP B.V. (NL) 2016-12-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10315996-B2 ROR gamma (RORγ) modulators RORA, RORB, RORC ABL1 2175/4885RIN1 1031/4885RORC 3/4885
US-20180170877-A1 ROR GAMMA (RORY) MODULATORS RORA, RORB, RORC ABL1 2035/4885RIN1 1084/4885RORC 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.