SCHEMBL18291376

SCHEMBL18291376

Nc1ccc(CC(=O)N2CCNC3(CC3)C2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46
GABRE P78334 1/20 0.46
GABRA6 Q16445 1/20 0.46
GABRG1 Q8N1C3 1/20 0.46
GABRG3 Q99928 1/20 0.46
GABRQ Q9UN88 1/20 0.46
NAMPT P43490 1/20 0.42
CPB1 P15086 3/20 0.38
HSD11B1 P28845 2/20 0.37
CRBN Q96SW2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20038221 0.86 HSD11B1 (0.37) HSD11B1CRBNCDK4SCN9AECE2
SCHEMBL20038223 0.86 VNN1 (0.39) HSD11B1CDK4SCN9AMC4RGHSR
SCHEMBL13768896 0.86 CDK4 (0.47) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL18291302 0.83 PANK3 (0.51) HSD11B1CDK4SCN9AMC4RGHSR
SCHEMBL20249346 0.83 PANK3 (0.37) HSD11B1CDK4SCN9AMC4RGHSR
SCHEMBL14084729 0.76 GABRP (0.58) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL18291431 0.76 IDH1 (0.37) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL2234473 0.73 MAPT (0.56) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL13769030 0.68 GABRP (0.48) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL18191789 0.68 GABRP (0.43) GABRPGABRDGABRA1GABRB1GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016194831-A1 PYRIDO[3,4-d]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 帝人ファーマ株式会社 2016-12-08 WO disclosed