SCHEMBL18308447

SCHEMBL18308447

COc1cc2c(c(N)c1C(N)=O)OCCO2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.48
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 4/20 0.46
POLB P06746 4/20 0.46
TDP1 Q9NUW8 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
LMNA P02545 3/20 0.40
HSD17B10 Q99714 1/20 0.40
CTNNB1 P35222 2/20 0.39
WNT3A P56704 2/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
TSHR P16473 2/20 0.37
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18308451 0.88 KDM4E (0.49) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL11982142 0.76 PLK1 (0.69) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL15988852 0.75 PLK1 (0.49) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL15988858 0.70 PLK1 (0.45) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL9110788 0.70 ALDH1A1 (0.51) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL14099207 0.70 PLK1 (0.47) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL16703478 0.69 LMNA (0.44) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL12184928 0.69 PLK1 (0.53) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL4715766 0.68 PLK1 (0.71) PLK1KDM4EALDH1A1POLBTDP1
SCHEMBL30330021 0.68 PLK1 (0.71) PLK1KDM4EALDH1A1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016199943-A1 HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-12-15 WO disclosed