SCHEMBL18315532

SCHEMBL18315532

Nc1ccc(C(=O)N2CC3(CCN(C(=O)O)CC3)C2)cc1O

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 5/20 0.63
ATXN2 Q99700 5/20 0.63
CYP3A4 P08684 4/20 0.42
GPR183 P32249 3/20 0.42
USP2 O75604 3/20 0.42
ALDH1A1 P00352 3/20 0.42
CYP2D6 P10635 3/20 0.42
HIF1A Q16665 2/20 0.42
CYP1A2 P05177 1/20 0.42
TSHR P16473 3/20 0.41
MAPK1 P28482 2/20 0.41
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23123044 0.80 ALDH1A1 (0.48) ENPP2ATXN2CYP3A4USP2ALDH1A1
SCHEMBL15540638 0.78 ENPP2 (1.00) ENPP2ATXN2
SCHEMBL18315558 0.77 CA12 (0.60) ENPP2ATXN2
SCHEMBL23123111 0.77 IP6K1 (0.43) ENPP2ATXN2CYP3A4USP2ALDH1A1
SCHEMBL15540286 0.77 ATXN2 (1.00) ENPP2ATXN2
SCHEMBL18315539 0.76 ENPP2 (0.58) ENPP2ATXN2CYP3A4USP2ALDH1A1
SCHEMBL23123113 0.76 USP2 (0.47) CYP3A4USP2ALDH1A1CYP2D6HIF1A
SCHEMBL5924169 0.75 HPGD (0.58) CYP3A4ALDH1A1CYP2D6CYP1A2TSHR
SCHEMBL5924363 0.74 HPGD (0.61) CYP3A4ALDH1A1CYP2D6CYP1A2TSHR
SCHEMBL15541236 0.73 ENPP2 (0.60) ENPP2ATXN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861566-B1 NEW DIAZASPIROCYCLOALKANE AND AZASPIROCYCLOALKANE HOFFMANN LA ROCHE (CH) 2016-12-21 EP claimed