SCHEMBL18322752

SCHEMBL18322752

Cc1nc(C2CCOCC2)c[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.37
HTR6 P50406 1/20 0.33
TDP2 O95551 1/20 0.33
PIK3CD O00329 3/20 0.33
PIK3CA P42336 1/20 0.33
PDE1B Q01064 1/20 0.33
DAO P14920 1/20 0.33
IRAK4 Q9NWZ3 3/20 0.32
CFTR P13569 1/20 0.32
MAPK1 P28482 1/20 0.32
MAPK8 P45983 1/20 0.31
MAPK9 P45984 1/20 0.31
MAPK10 P53779 1/20 0.31
CNR2 P34972 1/20 0.31
CHRNA7 P36544 1/20 0.31
MAP3K12 Q12852 2/20 0.31
CHEK1 O14757 1/20 0.31
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
PIK3CB P42338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19485454 0.81 HRH4 (0.37)
SCHEMBL3391231 0.81 HRH4 (0.37)
Hydrochloric Acid SCHEMBL947812 0.78 HRH4 (0.42) MAP3K12
SCHEMBL23123541 0.77 HTR6 (0.36) KDM5BHTR6PIK3CDPIK3CADAO
SCHEMBL22632160 0.76 HTR1D (0.42)
SCHEMBL18322564 0.75 TRPV3 (0.34) MAPK1
SCHEMBL7906841 0.70 TDP2 (0.33) KDM5BTDP2PDE1BDAOIRAK4
SCHEMBL21193094 0.70 CHRM2 (0.43) MAP3K12CHEK1
SCHEMBL23123505 0.68 F2 (0.34) HTR6IRAK4MAP3K12
SCHEMBL22632134 0.68 ENPP3 (0.35) KDM5BHTR6TDP2PIK3CDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307739-A1 NRF2 REGULATORS GlaxoSmithKline Intellectual Property Development Limited (GB) 2018-04-18 EP disclosed
WO-2016202253-A1 NRF2 REGULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2016-12-22 WO disclosed